Pembagian antibiotic berdasarkan daya ke
Pembagian antibiotic berdasarkan daya kerja
Bakteristatik mencegah dan
menghambat pertembuhan
kuman, tidak membunuhnya
sehingga pembasmiasn kuman
tergantung pada imunitas
1. Tetrasiklin
2. Spectinomicin
3. Sulphonamides
4. Macrolides
5. chlorampenicol
6. Trimetropin
Bakterisid à membasmi kuman
1. Penisilin
2. cephalosporin
3. fluorokuinolon(ciprofloxacin)
4. Monobactam
5. Carbapenem
6. Glycopeptida(vancomycin)
INHIBIT
CLASIFICATION
ANTIBIOTIK
Beta-lactamase
inhibit
sulbactam
Penicillins
Animopenicil
lin
(broad
spectrum)
Natural
penicillin
(narrow
spectrum)
Cephalosporin
Carbapenems
No
lactam
monobactams
glycopeptide
Other
Protein
30S Aminosynthesis
glycosides
DNA
Clavulanic tazobacta
Avibactam
acid
m
Penicinillase- sensible
Amphicilin
amoxicilin
Penicillin G: Na, K, procainic, benzathine(IV/IM)
Penicillin VK : VO
Penicinillase- resistance(very narrow spectrum)
Nafcilin
oxacillin
dicloxacillin
Antipseudomonal(extended spectrum)
carboxipenici ticarcillin
Carbenicillin
Piperacillin
llin
ureidopenicil azlocillin
mezlocillin
lin
First gene
cephalexine
cefazolin
cefadroxil
Cephradrine
cephapirin
Second gene
cefuroxime
cefprozil
cefaclor
cefoxitin
cefotetan
loracarbef
Third gene
cefoperazone
cefprozil
cefaclor
cefpodoxime
ceftrizoxime
cefotaxime
cefditoren
Fourth gene
cefepime
cefpirome
Fifth gene
ceftaroline
ceftolozane
Meropenem
Ertapenem
Doripenem
Imipenem+
cylastatine
Panipenem
Aztreonam
Tigemonam
Carumonam
Nocardinin A
vancomycin
Telavancin
Dalbavancin
Oritavancin
Colistin
Amikacin
Streptomycin
tetracyclins Doxycycline
tetracyclin
50S Oxazolidon Linezolid
ones
Streptogra quinupristin
minis
Chloramphenicol
Macrolides erythromycin
Lincosamid Clindamycin
es
Fluorquinolones
Ciprofloxacin
Polymycin B
Gentamicin
Daptomycin
Tobramycin
Neomycin
Minocycline
demeclocyli
Tigecyclin
azithromycin
Clarithromycin
lincomycin
Moxifloxacin
Levofloxacin
isoniazid
Gemifloxacin
topoisom
erase
quinolon
Folic acid Sulfonamides
synthesis
DHFR inhibitor
DNA
Nitroimidazoles
(Damage
)
mRNA
rifampim
synth.
Penicillin
Norfloxacin
Ofloxacin
Nalidixic acid
Sulfamethoxa Ag
zole(SMX)
sulfadiazine
Trimethropine(TMP)
Metronidazoles
Enofloxacin
Sparfloxacin
sulfasalazine
sulfisoxazole
Pyrimethamine
Tinidazole
AB
Dosis dewasa
Dosis anak
Penisilin G
Cara
pemberian
IV
1-4 mU/4-6j
Penisilin VK
PO
0,25-0,5 g qid
25.000400.000
unit/kg/h/46 dosis
25-50
mg/kg/h/4
dosis
Penisilin antistafilokokus
Kloksasilin
PO
dikloksasilin
0,25-0,5 g qid
Oksasilin
1-2g/4-6 j
IV
Penisilin yang diperluas
Amoksisilin
PO
0,25-0,5 g qid
Amoksisilin/as
. klavulanat
PO
Piperasilin
IV
500/125875/125 mg
bid-tid
3-4g/4-6 j
Tikarsilin
IV
3g/4-6 j
Panduan dosis sefalosforin
AB
Cara
pemberian
First gene
Cefadroxil
PO
cefeleksin
Dosis
neonates
75.000150.000
unit/kg/h/23 dosis
25-50
mg/kg/h/4
dosis
50-100
mg/kg/h/4-6
dosis
50-75
mg/kg/h/2-3
dosis
20-40
mg/kg/h/3
dosis
20-40
mg/kg/h/3
dosis
300
mg/kg/h/4-6
dosis
300
mg/kg/h/4-6
dosis
150
mg/kg/h/2
dosis
150-200
mg/kg/h/2-3
dosis
Dosis dewasa
Dosis anak
0,5-1 g/h-2x
30
mg/kg/h/2
dosis
Dosis
neonatus
Bakteristatik mencegah dan
menghambat pertembuhan
kuman, tidak membunuhnya
sehingga pembasmiasn kuman
tergantung pada imunitas
1. Tetrasiklin
2. Spectinomicin
3. Sulphonamides
4. Macrolides
5. chlorampenicol
6. Trimetropin
Bakterisid à membasmi kuman
1. Penisilin
2. cephalosporin
3. fluorokuinolon(ciprofloxacin)
4. Monobactam
5. Carbapenem
6. Glycopeptida(vancomycin)
INHIBIT
CLASIFICATION
ANTIBIOTIK
Beta-lactamase
inhibit
sulbactam
Penicillins
Animopenicil
lin
(broad
spectrum)
Natural
penicillin
(narrow
spectrum)
Cephalosporin
Carbapenems
No
lactam
monobactams
glycopeptide
Other
Protein
30S Aminosynthesis
glycosides
DNA
Clavulanic tazobacta
Avibactam
acid
m
Penicinillase- sensible
Amphicilin
amoxicilin
Penicillin G: Na, K, procainic, benzathine(IV/IM)
Penicillin VK : VO
Penicinillase- resistance(very narrow spectrum)
Nafcilin
oxacillin
dicloxacillin
Antipseudomonal(extended spectrum)
carboxipenici ticarcillin
Carbenicillin
Piperacillin
llin
ureidopenicil azlocillin
mezlocillin
lin
First gene
cephalexine
cefazolin
cefadroxil
Cephradrine
cephapirin
Second gene
cefuroxime
cefprozil
cefaclor
cefoxitin
cefotetan
loracarbef
Third gene
cefoperazone
cefprozil
cefaclor
cefpodoxime
ceftrizoxime
cefotaxime
cefditoren
Fourth gene
cefepime
cefpirome
Fifth gene
ceftaroline
ceftolozane
Meropenem
Ertapenem
Doripenem
Imipenem+
cylastatine
Panipenem
Aztreonam
Tigemonam
Carumonam
Nocardinin A
vancomycin
Telavancin
Dalbavancin
Oritavancin
Colistin
Amikacin
Streptomycin
tetracyclins Doxycycline
tetracyclin
50S Oxazolidon Linezolid
ones
Streptogra quinupristin
minis
Chloramphenicol
Macrolides erythromycin
Lincosamid Clindamycin
es
Fluorquinolones
Ciprofloxacin
Polymycin B
Gentamicin
Daptomycin
Tobramycin
Neomycin
Minocycline
demeclocyli
Tigecyclin
azithromycin
Clarithromycin
lincomycin
Moxifloxacin
Levofloxacin
isoniazid
Gemifloxacin
topoisom
erase
quinolon
Folic acid Sulfonamides
synthesis
DHFR inhibitor
DNA
Nitroimidazoles
(Damage
)
mRNA
rifampim
synth.
Penicillin
Norfloxacin
Ofloxacin
Nalidixic acid
Sulfamethoxa Ag
zole(SMX)
sulfadiazine
Trimethropine(TMP)
Metronidazoles
Enofloxacin
Sparfloxacin
sulfasalazine
sulfisoxazole
Pyrimethamine
Tinidazole
AB
Dosis dewasa
Dosis anak
Penisilin G
Cara
pemberian
IV
1-4 mU/4-6j
Penisilin VK
PO
0,25-0,5 g qid
25.000400.000
unit/kg/h/46 dosis
25-50
mg/kg/h/4
dosis
Penisilin antistafilokokus
Kloksasilin
PO
dikloksasilin
0,25-0,5 g qid
Oksasilin
1-2g/4-6 j
IV
Penisilin yang diperluas
Amoksisilin
PO
0,25-0,5 g qid
Amoksisilin/as
. klavulanat
PO
Piperasilin
IV
500/125875/125 mg
bid-tid
3-4g/4-6 j
Tikarsilin
IV
3g/4-6 j
Panduan dosis sefalosforin
AB
Cara
pemberian
First gene
Cefadroxil
PO
cefeleksin
Dosis
neonates
75.000150.000
unit/kg/h/23 dosis
25-50
mg/kg/h/4
dosis
50-100
mg/kg/h/4-6
dosis
50-75
mg/kg/h/2-3
dosis
20-40
mg/kg/h/3
dosis
20-40
mg/kg/h/3
dosis
300
mg/kg/h/4-6
dosis
300
mg/kg/h/4-6
dosis
150
mg/kg/h/2
dosis
150-200
mg/kg/h/2-3
dosis
Dosis dewasa
Dosis anak
0,5-1 g/h-2x
30
mg/kg/h/2
dosis
Dosis
neonatus