Formulasi dan Evaluasi Pemakaian Cangkang Kapsul Alginat untuk Pembuatan Sediaan Floating dari Dispersi Padat Aspirin

DAFTAR PUSTAKA
Abdou, H.M., Samir, H., dan Naseem, M. (2001). Dissolution. Dalam:
Remington: The Science and Practice of Pharmacy. Volume 1. Editor
Alfonso R. Gennaro. Philadelphia: Lipincott Williams and Wilkins.
Halaman 654.
Ansel, H. C. (2005). Pengantar Bentuk Sediaan Farmasi. Edisi keempat. Jakarta:
UI Press. Halaman 217-218.
Arunachalam, A., Karthikeyen, M., Kishore, K., Pottabathula, H. P., Sethurman,
S., Ashutoshkumar, S., dan Manidipa, S. Floating Drug Delivery System:
A review. International Journal of Research in Pharmaceutical Sciences .
2(1): 77.
Atkins, P.W. (1999). Kimia Fisika . Jilid Ketiga. Jakarta: Erlangga. Halaman 169.
Attwood, D., dan Florence, A. T. (2008). Physical Pharmacy. London:
Pharmaceutical Press. Halaman 89.
Bangun, H., Simanjuntak, M. T., Tarigan, P., dan Ismanelly, T. (2005).
Pembuatan dan Karakterisasi Kapsul Alginat yang Tahan terhadap Asam
Lambung. Media Farmasi. 13(1): 70-79.
Bangun, H. (2002). The Preparation of Indomethacin Capsules Without
Gastrointestinal Side Effect. The 32 nd Korean Society Annual Meeting
Pharmaceutics in Asia . 28-29 November.
Belitz, H. D., Grosch, W., dan Schieberle, P. (2009). Food Chemistry. Edisi

Keempat. Berlin: Springer-Verlag. Halaman 232.
Berardi, R.R., dan Welage, L. S. (2005). Peptic Ulcer Disease . Dalam:
Pharmacotherapy: A Pathopysiologic Approach. Edisi Keenam. Editor
Joseph T. Dipiro. New York: McGraw-Hill. Halaman 630.
Chhater, S., dan Praveen, K. (2013). Solvent Evaporation Method for Amorphous
Solid Dispersion: Predictive Tools for Improve The Dissolution Rate of
Pioglitazone Hydrochloride. International Journal of Pharmaceutical
Chemical and Biological Sciences . 3(2): 350-359.
Chiou, W.L., dan Riegelman, S. (1971). Pharmaceutical Application of Solid
Dispersion System. Journal of Pharmaceutical Science. 60(9): 81-94.
Corwin, E.J. (2009). Buku Saku Patofisiologi. Edisi Ketiga. Jakarta: Penerbit
Buku Kedokteran EGC. Halaman 603-605.
Craig, D.Q.M. (2002). The Mechanisms of Drug Release From Solid Dispersion
in Water-Soluble Polymers. Int. J. Pharm. 24(3): 131-144.

66
Universitas Sumatera Utara

Dewoto, H. R. (2008). Antikoagulan, Antitrombotik, Trombolitik dan Hemostatik:
Farmakologi dan Terapi. Edisi kelima. Jakarta: Balai Penerbit FK UI.

Halaman 804-819.
Dey, S., dan Saha, P. (2013). Floating Drug Delivery System. International
Journal of Pharmacy and Engineering (IJPE) . 1(1): 3-4.
Ditjen POM. (1995). Farmakope Indonesia . Edisi Keempat. Jakarta: Depkes RI.
Halaman 34.
Dwivedi, S., dan Kumar, V. (2011). Floating Drug Delievery System – A Concept
of Gastroretention Dosages Form. International Journal of Research in
Pharmaceutical and Biomedical Sciences . 2(4): 1413-1414.
Draget, K.I., Smidsrod, O., dan Gudmund S. (2005). Alginate from Algae .
Weinheim: WILEY-VCH Verlag GmbH and Co. Halaman 3-4.
Gennaro, R.A. (2000). Remington: The Science and Practice of Pharmacy. Edisi
ke-20. New York. Lippincott Williams & Wilkins. Halaman 885.
Goldberg, A. H., Gibaldi, M., Kanig, J. L. (1966). Increasing dissolution rates and
gastrointestinal absorption of drug via solid solutions and eutectic mixtures
II. Experimental evaluation of a eutectic mixture: urea-acetaminophen
system. J Pharm Sci. 1-3.
Gopalakrishnan, S., dan Chenthilnathan, A. (2011). Floating Drug Delivery
Systems: A Review. Journal of Pharmaceutical Science and Technology.
3(2): 548-554.
Goyal., M., Rajesh, P., Kapil, K. P., dan Mehta, S. C. (2011). Floating Drug

Delivery System. Journal of Current Pharmaceutical Research .
5(1): 7-18.
Itai, S. N. M., Kouchiwa, S., Muraysma, H., Nagai, T. (1985). Influence of
wetting factors on the dissolution behavior of fufenamic acid. Chem
Pharm: Bull. 64-73.
Hascicek, C., Turkmen, G., Ozdemir, N., dan Tilkan, G. Y. (2011). Effect of
formulation parameters on the drug release and floating properties of
gastric floating two-layer tablets with acetylsalicylic acid. Ankara: Acta
Pharm. 61: 303-312.
Knight, J.C. (2003). Antiplatelet Treatment in Stable Coronary Artery Disease.
Heart. 89: 1273-1278.
Kumar, S. K. P., Bhowmik, D., dan Srivastava, S. (2012). Sustained Release Drug
Delivery System Potential. 1(2): 46-48.
Lachman, L., Liebermen, H. A., dan Kanig, J. L. (2008). Teori dan Praktek
Farmasi Industri II . Edisi ketiga. Jakarta: UI-Press. Halaman 834-837.

67
Universitas Sumatera Utara

Lanza, F.L. (1988). A Review of Gastric Ulcer and Gastroduodenal Injury in

Normal Volunteers Receiving Aspirin and Other Non-Steroidal AntiInflamatory Drugs. Scan J Gastroentol. 24(163): 24-31.
Leeson, C.R., Thomas, S.L., dan Anthony, A.P. (1989). Buku Ajar Histology. Alih
Bahasa: dr. Yan Tambayong. Jakarta: Penerbit Buku kedokteran EGC.
Halaman 347-357.
Leuner, C., dan Dressman, J. (2002). Improving Drug Solubility For Oral
Delivery Using Solid Dispersion. Eur. J. Pharm. Biopharm. 40(7): 47-60.
Levy, G. (1963). Effect of Particle Size on Dissolution and Gastrointestinal
Absorption Rates of Pharmaceuticals. Am. J. Pharm. 135: 78-92.
Martin, A., Swarbrik, J., dan Cammarata, A. (2008). Dasar –dasar Farmasi Fisik
dalam Ilmu Farmasetik. Alih Bahasa Yoshita. Edisi Ketiga. Jakarta: UI
Press. Halaman 1170-1171, 1174.
Morris, E.R., Rees, D. A., dan Thom, D. (1980). Characterisation of Alginates
Composition and Block Structure by Circular Dichroism. Carbohydrate
Research . 81(2): 305-310.
Mycek, M.J., Harver, R. A., dan Champe, P. C. (2001). Farmakologi Ulasan
Bergambar . Jakarta: Widya Medika. Halaman 196-199.
Narang, N. (2011). An Updated Review On: Floating Drug Delivery System
(FDDS). International Journal of Applied Pharmaceutics. 3(1): 2-4.
Nayak, A. K., Maji, R., dan Das, B. (2010). Gastroretentive Drug Delivery
Systems: a review. Asian Journal of Pharmaceutical and Clinical

Research . 3(1): 3-4.
Pawar, V. K., Kansal, S., Garg, G., Awasthi, R., Singodia, D., dan Kulkarni, G. T.
(2011). Gastroretentive Dosage Forms: A Review with Special Emphasis
on Floating Drug Delivery Systems. Drug Deliv. 18: 97-110
Price, S. A., dan Wilson, L. M. (1995). Patofisiologi: Konsep Klinis Prosesproses Penyakit. Volume 1. Edisi keempat. Jakarta: Penerbit Buku
Kedokteran EGC. Halaman 423-430.
Shargel, L., dan Andrew, A. (1998). Biofarmasetika dan Farmakokinetika
Terapan . Penerjemah: Fasich dan Siti Sjamsijah. Edisi Kedua. Surabaya:
Airlangga University Press. Halaman 86-112.
Sharma, S.,dan Garg, S. (2003). Gastroretentive Drug Delivery System in Drug
Delivery Oral. Business Brief: Pharmatech . Halaman 160-166.
Sharma, N., Dilip, A., Gupta, M. K., dan Mahaveer, P. K. (2011). A
Comprehensive Review on Floating Drug Delivery System. International

68
Universitas Sumatera Utara

Journal of Research in Pharmaceutical and Biomedical Sciences .
2(2): 428-429.


Shiraishi, S., Imai, T., Iwaoka, D., dan Otagiri. (1991). Improvement of
Absorption Rate of Indomethacin and Reduction of Stomach Irritation by
Alginate Dispersion. J.Pharm.Pharmacol. 43: 615-620.
Simamora, E.R.F. (2014). Studi Pemakaian Cangkang Kapsul Alginat sebagai
Sediaan Floating dari Metronidazol. Program Studi Ilmu Farmasi.
Program Sarjana Universitas Sumatera Utara. Medan.
Simonelli, A.P., Mehta, S.C., dan Higuchi, W.I. (1969). Dissolution Rates of High
Energy Polyvinylpyrrolidone (PVP) - Sulphathiazole Coprecipitates. J.
Pharm. Sci. 58: 538-549.
Sinurat, D. (2005). Studi Pelepasan Ketersediaan Hayati dan Efek Iritasi
Terhadap Lambung dari Kapsul Alginat yang Mengandung Aspirin
Dibandingkan dengan Tablet Salut Enterik yang Beredar di Perdagangan .
Program Studi Ilmu Farmasi. Program Pasca Sarjana Universitas Sumatera
Utara. Medan.
Smallman, R.E. (2000). Metalurgi Fisik Modern dan Rekayasa Material . Jakarta:
Erlangga. Halaman 146-147.
Soppimath, K.S., Kulkarni, A.R., Rudzinski, W.E., dan Aminabhavi, T.M. (2001).
Microspheres As Floating Drug Delivery Systems to Increase Gastric
Retention of Drugs. Drug Metab Rev. 33: 149-160.
Sunil, K., Amandeep, K., Robin, S., dan Ramica, S. (2012). Peptic Ulcer: A

Review on Etiology and Pathogenesis. International Research Journal of
Pharmacy. 3(6): 1-2.
Tan, H. T., dan Rahardja, K. (2003). Obat-obat penting . Edisi kelima. Cetakan
Kedua. Jakarta: PT. Elex Media Komputindo. Halaman 181-182.
Thom, D., Toft, K., dan Walsh, M. J. (1980). Interchain Associations of Alginates
and Pectins. Program Food Nutrition Science . 6(8): 97-108.
Wilmana, P.F. (1995). Analgesik-Antipiretik, Antiinflamasi Nonsteroid dan Obat
Pirai: Farmakologi dan Terapi. Edisi keempat. Jakarta: Bagian
Farmakologi Fakultas Kedokteran Universitas Indonesia. Halaman 218.
Zhanjiang, F. (1990). Training Manual of Gracilaria Culture and Seaweed
Proscessing in China . Regional Seafarming Development and
Demonstration Project China. http://www.fao.org/docrep/fi eld/003 ab
730e/.htm . Diunduh pada tanggal 23 Juli 2014

69
Universitas Sumatera Utara